Emijoy DS Tablet

Chlordiazepoxide
25 mg + 10 Mg
Beximco Pharmaceuticals Ltd.
Pack size 30's pack
Dispensing mode
Source
Agent
Retail Price 12.00 AED

Indications

Emijoy DS Tablet is used for: Anxiety, Insomnia, Muscle spasms, Acute symptoms of alcohol withdrawal

Adult Dose

Oral Insomnia Adult: 10-30 mg before bedtime. Muscle spasms Adult: 10-30 mg daily in divided doses. Anxiety Adult: 30 mg daily in divided doses, up to 100 mg daily in severe conditions. Acute symptoms of alcohol withdrawal Adult: 25-100 mg daily repeated as necessary. Max dose: 300 mg daily.

Child Dose

Anxiety <6 years: Safety and efficacy not established >6 years: 0.5 mg/kg/day divided PO q6-8hr, OR 5 mg PO q6-12hr; may increase dose to 10 mg PO q8-12hr

Renal Dose

Renal impairment CrCl <10 mL/min: 50% of recommended dose CrCl >10 mL/min: Dose adjustment not necessary (monitor)

Administration

May be taken with or without food.

Contra Indications

Acute pulmonary insufficiency, resp depression, patients with marked neuromuscular resp weakness; hypersensitivity to benzodiazepines; chronic psychosis; porphyria; pregnancy and lactation.

Precautions

Concomitant use of benzodiazepines and opioids may result in profound respiratory depression, coma, and death; administer concomitantly when there are no alternative options; limit dosages and durations to minimum required; monitor for signs and symptoms of respiratory depression and sedation Addiction, abuse, and misuse On September 2020, FDA addressed serious risks of benzodiazepine addiction, abuse, and misuse, which can lead to overdose and death Physical dependence can occur when taken steadily for several days to weeks, even as prescribed Stopping abruptly or reducing dosage too quickly can result in withdrawal reactions, including seizures, which can be life-threatening Assess each patient’s risk prior to prescribing and monitor regularly for the development of these behaviors or conditions Patient should be observed for up to 3 hours following administration Anterograde amnesia associated with treatment Use caution in renal and hepatic impairment Use caution in respiratory disease (COPD), sleep apnea, porphyria, open-angle glaucoma (questionable), depression, suicidal ideation, impaired gag reflex May impair ability to perform hazardous tasks Paradoxical reactions, including hyperactive or aggressive behavior, reported Use caution in patients with depression, especially if suicidal risk present Ataxia and oversadation may occur in the elderly and debilitated patients; there also increased risk of falls Use caution in patients with history of drug abuse or acute alcoholism; tolerance, psychological and physical dependence may occur with prolonged use

Pregnancy-Lactation

Pregnancy category: D Lactation: Enters breast milk/not recommended

Interactions

Cimetidine increases serum conc of chlordiazepoxide. Potentiates the action of major neuroleptics. The concomitant use of benzodiazepines and opioids increases the risk of respiratory depression because of actions at different receptor sites in the CNS that control respiration. Benzodiazepines interact at GABAA sites and opioids interact primarily at mu receptors. When benzodiazepines and opioids are combined, the potential for benzodiazepines to significantly worsen opioid-related respiratory depression exists. Limit dosage and duration of concomitant use of benzodiazepines and opioids, and monitor patients closely for respiratory depression and sedation. Potentially Fatal: Alcohol potentiates CNS-depressant effect of chlordiazepoxide. Contraindicated (0) Serious (33) apalutamide benzhydrocodone/acetaminophen buprenorphine subdermal implant buprenorphine transdermal buprenorphine, long-acting injection calcium/magnesium/potassium/sodium oxybates conivaptan dacomitinib enzalutamide fentanyl fentanyl intranasal fentanyl iontophoretic transdermal system fentanyl transdermal fentanyl transmucosal fexinidazole hydrocodone idelalisib ivosidenib lonafarnib methohexital metoclopramide intranasal nefazodone oliceridine olopatadine intranasal opicapone remifentanil selinexor sodium oxybate sufentanil SL tolcapone tucatinib valerian zuranolone

Adverse Effects

Side effects of Chlordiazepoxide : >10% Ataxia,Drowsiness,Memory impairment,Sedation,Muscle weakness,Rash,Decreased libido,Menstrual disorders,Xerostomia,Salivation decreased,Increased/decreased appetite,Weight gain/loss,Micturition difficulties 1-10% Confusion,Dizziness,Disinhibition,Akathisia,Dermatitis,Hypotension,Salivation increased,Sexual dysfunction,Incontinence,Rigidity,Tremor,Muscle cramps,Tinnitus,Nasal congestion

Mechanism of Action

Chlordiazepoxide enhances activity of the inhibitory transmitter GABA in different parts of CNS by increasing neuronal-membrane permeability to chloride ions resulting to hyperpolarisation and stabilisation. It has some muscle relaxant and anticonvulsant activity.

Note

Emijoy DS 25 mg + 10 Mg Tablet manufactured by Beximco Pharmaceuticals Ltd.. Its generic name is Chlordiazepoxide. Emijoy DS is availble in Bangladesh. Farmaco BD drug index information on Emijoy DS Tablet is not intended for diagnosis, medical advice or treatment; neither intended to be a substitute for the exercise of professional judgment.

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